1138245-21-2 structure, C18H25NO5S

Mirogabalin besylate

CAS No.

1138245-21-2

Formula:

C18H25NO5S

Basic Info

Mirogabalin (DS-5565) is a drug developed by Daiichi Sankyo and related to drugs such as gabapentin and pregabalin. Similarly to these drugs, mirogabalin binds to the α2δ calcium channels (1 and 2), but with significantly higher potency than pregabalin. It has shown promising results in Phase II clinical trials for the treatment of diabetic peripheral neuropathic pain, and is currently in Phase III trials.

Formula
C18H25NO5S
Molecular Weight
367.46
Exact Mass
367.145
LogP
4.4968
PSA
126.07
Synonyms

DS-5565 besylate

[(1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid benzenesulfonate

[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid monobenzenesulfonate

expand collapse

Related Compound Information